Class information for:
Level 1: PROCATEROL//AGONIST ANTAGONIST DISCRIMINATION//BROXATEROL

Basic class information

Class id #P Avg. number of
references
Database coverage
of references
31281 155 24.0 43%



Bar chart of Publication_year

Last years might be incomplete

Hierarchy of classes

The table includes all classes above and classes immediately below the current class.



Cluster id Level Cluster label #P
0 4 BIOCHEMISTRY & MOLECULAR BIOLOGY//CELL BIOLOGY//ONCOLOGY 4064930
54 3       ASTHMA//RESPIRATORY SYSTEM//ALLERGY 90590
397 2             ASTHMA//JOURNAL OF ASTHMA//INHALED CORTICOSTEROIDS 16767
31281 1                   PROCATEROL//AGONIST ANTAGONIST DISCRIMINATION//BROXATEROL 155

Terms with highest relevance score



rank Term termType Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 PROCATEROL authKW 547217 6% 28% 10
2 AGONIST ANTAGONIST DISCRIMINATION authKW 443256 2% 75% 3
3 BROXATEROL authKW 295502 2% 50% 3
4 THERMODYNAMIC DISCRIMINATION authKW 262670 1% 67% 2
5 8 OH DPAT WAY 100135 authKW 197003 1% 100% 1
6 AGONISM ANTAGONISM authKW 197003 1% 100% 1
7 AGONIST AND ANTAGONIST DISCRIMINATION authKW 197003 1% 100% 1
8 ANTAGONIST BINDING ENTHALPIES authKW 197003 1% 100% 1
9 ATRIAL BEATS authKW 197003 1% 100% 1
10 BETA 2 ADRENOCEPTOR SELECTIVE AGONISTS authKW 197003 1% 100% 1

Web of Science journal categories



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 Pharmacology & Pharmacy 1601 59% 0% 91
2 Allergy 560 9% 0% 14
3 Respiratory System 119 8% 0% 12
4 Chemistry, Medicinal 88 8% 0% 12
5 Medicine, Research & Experimental 40 7% 0% 11
6 Social Sciences, Interdisciplinary 31 3% 0% 4
7 Integrative & Complementary Medicine 3 1% 0% 1
8 Immunology 2 4% 0% 6
9 Toxicology 2 2% 0% 3
10 Mathematics, Interdisciplinary Applications 2 1% 0% 2

Address terms



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 FARMAKOL TER EUT 197003 1% 100% 1
2 PHARMACEUT CHEM CO DD 197003 1% 100% 1
3 CHAIR PHARMACOL MED 98501 1% 50% 1
4 NEW PROD EVALUAT DEV 98501 1% 50% 1
5 SHINANOZAKA CLIN 98501 1% 50% 1
6 CLIN EXPT MEDPHARMACOL UNIT 49249 1% 25% 1
7 MORPHOL HISTOL 49247 1% 13% 2
8 CLIN STUDY UNIT 39399 1% 20% 1
9 NAZL ECCELLENZA SVILUPPO METODOL INNOVAT STUD 32832 1% 17% 1
10 RACEHORSE HOSP 28142 1% 14% 1

Journals



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 ANNALS OF ALLERGY 5393 5% 0% 8
2 INTERNATIONAL JOURNAL OF CLINICAL PHARMACOLOGY RESEARCH 3286 3% 0% 4
3 BIOCHEMICAL PHARMACOLOGY 2083 9% 0% 14
4 INTERNATIONAL JOURNAL OF CLINICAL PHARMACOLOGY AND THERAPEUTICS 1814 4% 0% 6
5 JOURNAL OF CLINICAL IMMUNOASSAY 1525 1% 1% 1
6 CURRENT CONTENTS/LIFE SCIENCES 1277 1% 0% 2
7 CURRENT THERAPEUTIC RESEARCH-CLINICAL AND EXPERIMENTAL 1022 3% 0% 5
8 EUROPEAN JOURNAL OF PHARMACOLOGY 1000 8% 0% 12
9 CURRENT CONTENTS/CLINICAL MEDICINE 919 1% 0% 1
10 RESPIRATION 877 3% 0% 4

Author Key Words



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
LCSH search Wikipedia search
1 PROCATEROL 547217 6% 28% 10 Search PROCATEROL Search PROCATEROL
2 AGONIST ANTAGONIST DISCRIMINATION 443256 2% 75% 3 Search AGONIST+ANTAGONIST+DISCRIMINATION Search AGONIST+ANTAGONIST+DISCRIMINATION
3 BROXATEROL 295502 2% 50% 3 Search BROXATEROL Search BROXATEROL
4 THERMODYNAMIC DISCRIMINATION 262670 1% 67% 2 Search THERMODYNAMIC+DISCRIMINATION Search THERMODYNAMIC+DISCRIMINATION
5 8 OH DPAT WAY 100135 197003 1% 100% 1 Search 8+OH+DPAT+WAY+100135 Search 8+OH+DPAT+WAY+100135
6 AGONISM ANTAGONISM 197003 1% 100% 1 Search AGONISM+ANTAGONISM Search AGONISM+ANTAGONISM
7 AGONIST AND ANTAGONIST DISCRIMINATION 197003 1% 100% 1 Search AGONIST+AND+ANTAGONIST+DISCRIMINATION Search AGONIST+AND+ANTAGONIST+DISCRIMINATION
8 ANTAGONIST BINDING ENTHALPIES 197003 1% 100% 1 Search ANTAGONIST+BINDING+ENTHALPIES Search ANTAGONIST+BINDING+ENTHALPIES
9 ATRIAL BEATS 197003 1% 100% 1 Search ATRIAL+BEATS Search ATRIAL+BEATS
10 BETA 2 ADRENOCEPTOR SELECTIVE AGONISTS 197003 1% 100% 1 Search BETA+2+ADRENOCEPTOR+SELECTIVE+AGONISTS Search BETA+2+ADRENOCEPTOR+SELECTIVE+AGONISTS

Core articles

The table includes core articles in the class. The following variables is taken into account for the relevance score of an article in a cluster c:
(1) Number of references referring to publications in the class.
(2) Share of total number of active references referring to publications in the class.
(3) Age of the article. New articles get higher score than old articles.
(4) Citation rate, normalized to year.



Rank Reference # ref.
in cl.
Shr. of ref. in
cl.
Citations
1 MERIGHI, S , SIMIONI, C , GESSI, S , VARANI, K , BOREA, PA , (2010) BINDING THERMODYNAMICS AT THE HUMAN CANNABINOID CB1 AND CB2 RECEPTORS.BIOCHEMICAL PHARMACOLOGY. VOL. 79. ISSUE 3. P. 471 -477 18 72% 7
2 HISHINUMA, S , SUGAWARA, K , UESAWA, Y , FUKUI, H , SHOJI, M , (2014) DIFFERENTIAL THERMODYNAMIC DRIVING FORCE OF FIRST- AND SECOND-GENERATION ANTIHISTAMINES TO DETERMINE THEIR BINDING AFFINITY FOR HUMAN H-1 RECEPTORS.BIOCHEMICAL PHARMACOLOGY. VOL. 91. ISSUE 2. P. 231 -241 19 51% 0
3 GILLI, P , FERRETTI, V , GILLI, G , BOREA, PA , (1994) ENTHALPY-ENTROPY COMPENSATION IN DRUG-RECEPTOR BINDING.JOURNAL OF PHYSICAL CHEMISTRY. VOL. 98. ISSUE 5. P. 1515-1518 13 46% 160
4 HARPER, EA , BLACK, JW , (2007) HISTAMINE H-3-RECEPTOR AGONISTS AND IMIDAZOLE-BASED H-3-RECEPTOR ANTAGONISTS CAN BE THERMODYNAMICALLY DISCRIMINATED.BRITISH JOURNAL OF PHARMACOLOGY. VOL. 151. ISSUE 4. P. 504-517 12 34% 6
5 CHETTA, A , GARAVALDI, G , CUOMO, A , GURRIERI, G , OLIVIERI, D , (1988) EARLY BRONCHODILATING EFFECT OF A NEW ORAL BETA-2-RECEPTOR AGONIST (BROXATEROL) IN BRONCHIAL-ASTHMA.RESPIRATION. VOL. 53. ISSUE 4. P. 220-224 9 90% 1
6 YU, TW , CHEN, RRL , GAU, CS , (2005) A NOVEL LIQUID CHROMATOGRAPHY/MASS/MASS SPECTROMETRY SYSTEM TO DETERMINE PROCATEROL LEVELS IN HUMAN PLASMA.JOURNAL OF FOOD AND DRUG ANALYSIS. VOL. 13. ISSUE 4. P. 312-318 5 83% 1
7 GILLI, P , GILLI, G , BOREA, PA , VARANI, K , SCATTURIN, A , DALPIAZ, A , (2005) BINDING THERMODYNAMICS AS A TOOL TO INVESTIGATE THE MECHANISMS OF DRUG-RECEPTOR INTERACTIONS: THERMODYNAMICS OF CYTOPLASMIC STEROID/NUCLEAR RECEPTORS IN COMPARISON WITH MEMBRANE RECEPTORS.JOURNAL OF MEDICINAL CHEMISTRY. VOL. 48. ISSUE 6. P. 2026 -2035 15 26% 12
8 BANERJEE, B , GANGULY, DK , (1996) THERMODYNAMICS OF THE INTERACTION OF D-TUBOCURARINE WITH NICOTINIC RECEPTORS OF MAMMALIAN SKELETAL MUSCLE IN VITRO.EUROPEAN JOURNAL OF PHARMACOLOGY. VOL. 310. ISSUE 1. P. 13-17 6 86% 6
9 KUSANO, K , NOMURA, M , TOJU, K , ISHIKAWA, Y , MINAMIJIMA, Y , YAMASHITA, S , NAGATA, S , (2016) PHARMACOKINETICS OF PROCATEROL IN THOROUGHBRED HORSES.JOURNAL OF VETERINARY PHARMACOLOGY AND THERAPEUTICS. VOL. 39. ISSUE 3. P. 264 -270 7 41% 0
10 MAGUIRE, PA , LOEW, GH , (1996) THERMODYNAMICS OF LIGAND BINDING TO THE CLONED DELTA-OPIOID RECEPTOR.EUROPEAN JOURNAL OF PHARMACOLOGY. VOL. 318. ISSUE 2-3. P. 505-509 8 62% 9

Classes with closest relation at Level 1



Rank Class id link
1 11521 OXITROPIUM BROMIDE//IPRATROPIUM BROMIDE//BERODUAL
2 17824 H 3ETORPHINE//H 3DIPRENORPHINE//SNPYS GROUP
3 33447 TULAREMIA LIVE VACCINE//ANTHRAX LIVE VACCINE//HEPATOMA H 2 73
4 25252 ISOTHERMAL TITRATION CALORIMETRY//ITC//CALORIMETRIC ENTHALPY
5 27138 1 OCTANOL WATER//OCTANOL WATER INTERFACE//UNSTIRRED LAYER THICKNESS
6 28500 3D NMR STRUCTURES//ACTH1 10//AMPHIPHILIC HELICAL PEPTIDE
7 32091 1 4 PERHYDROTHIAZINES//THIODIGLYCOL//2 METHOXYPHENYLMETYRAPONE
8 34996 ACTIVE CENTER ANALOGS OF SUPEROXIDE DISMUTASE//COFPLATON//COFPROPAMINE
9 29110 PLASMA EXUDATION//PLASMA PROTEIN EXUDATION//AIRWAY BARRIERS
10 7382 JOURNAL OF CYCLIC NUCLEOTIDE RESEARCH//JOURNAL OF CYCLIC NUCLEOTIDE AND PROTEIN PHOSPHORYLATION RESEARCH//JOURNAL OF RECEPTOR RESEARCH

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