Class information for:
Level 1: EXPLORATORY DISCOVERY//CYCLIC IMINES//3 ACYLLACTAMS

Basic class information

ID Publications Average number
of references
Avg. shr. active
ref. in WoS
29412 153 25.9 72%



Bar chart of Publication_year

Last years might be incomplete

Classes in level above (level 2)



ID, lev.
above
Publications Label for level above
2982 2124 ENDOCRINE POLYPEPTIDE CANC//LHRH RECEPTOR//SECT EXPT MED

Terms with highest relevance score



Rank Term Type of term Relevance score
(tfidf)
Class's shr.
of term's tot.
occurrences
Shr. of publ.
in class containing
term
Num. of
publ.
in class
1 EXPLORATORY DISCOVERY Address 11 69% 6% 9
2 CYCLIC IMINES Author keyword 2 23% 5% 7
3 3 ACYLLACTAMS Author keyword 1 100% 1% 2
4 NON PEPTIDE LHRH ANTAGONISTS Author keyword 1 100% 1% 2
5 C 14CARBON MONOXIDE Author keyword 1 50% 1% 1
6 MULTI WELL ASSAY Author keyword 1 50% 1% 1
7 OXIRANE 2 CARBOXAMIDES Author keyword 1 50% 1% 1
8 TRIAZINEDIONE Author keyword 1 50% 1% 1
9 TRIAZINETRIONE Author keyword 1 50% 1% 1
10 NON PEPTIDIC Author keyword 1 29% 1% 2

Web of Science journal categories

Author Key Words



Rank Web of Science journal category Relevance score
(tfidf)
Class's shr.
of term's tot.
occurrences
Shr. of publ.
in class containing
term
Num. of
publ.
in class
LCSH search Wikipedia search
1 CYCLIC IMINES 2 23% 5% 7 Search CYCLIC+IMINES Search CYCLIC+IMINES
2 3 ACYLLACTAMS 1 100% 1% 2 Search 3+ACYLLACTAMS Search 3+ACYLLACTAMS
3 NON PEPTIDE LHRH ANTAGONISTS 1 100% 1% 2 Search NON+PEPTIDE+LHRH+ANTAGONISTS Search NON+PEPTIDE+LHRH+ANTAGONISTS
4 C 14CARBON MONOXIDE 1 50% 1% 1 Search C+14CARBON+MONOXIDE Search C+14CARBON+MONOXIDE
5 MULTI WELL ASSAY 1 50% 1% 1 Search MULTI+WELL+ASSAY Search MULTI+WELL+ASSAY
6 OXIRANE 2 CARBOXAMIDES 1 50% 1% 1 Search OXIRANE+2+CARBOXAMIDES Search OXIRANE+2+CARBOXAMIDES
7 TRIAZINEDIONE 1 50% 1% 1 Search TRIAZINEDIONE Search TRIAZINEDIONE
8 TRIAZINETRIONE 1 50% 1% 1 Search TRIAZINETRIONE Search TRIAZINETRIONE
9 NON PEPTIDIC 1 29% 1% 2 Search NON+PEPTIDIC Search NON+PEPTIDIC
10 FISCHER REACTION 1 19% 2% 3 Search FISCHER+REACTION Search FISCHER+REACTION

Key Words Plus



Rank Web of Science journal category Relevance score
(tfidf)
Class's shr.
of term's tot.
occurrences
Shr. of publ.
in class containing
term
Num. of
publ. in
class
1 SUBSTITUTED INDOLE 5 CARBOXAMIDES 25 77% 11% 17
2 INDOLE 5 ACETAMIDES 15 77% 7% 10
3 2 3 5 DIMETHYLPHENYLTRYPTAMINE 11 100% 4% 6
4 2 ARYLINDOLES 11 69% 6% 9
5 LHRH ANTAGONISTS 9 67% 5% 8
6 IMIDAZOLO1 2 ALPHAPYRIMID 5 ONES 8 100% 3% 5
7 BENZIMIDAZOLE 5 SULFONAMIDES 6 80% 3% 4
8 NBI 42902 6 100% 3% 4
9 GNRH RECEPTOR ANTAGONISTS 3 42% 3% 5
10 H PROTECTING GROUP 2 67% 1% 2

Journals

Reviews



Title Publ. year Cit. Active references % act. ref.
to same field
Non-peptidic GnRH receptor antagonists 2004 18 45 69%
Nonpeptide gonadotropin releasing hormone antagonists 2004 11 41 88%
Recent advances in small molecule gonadotrophin-releasing hormone receptor antagonists 2004 13 19 79%
Non-peptide gonadotropin-releasing hormone receptor antagonists 2008 22 107 45%
G Protein-Coupled Receptors of the Hypothalamic-Pituitary-Gonadal Axis: A Case for GnRH, LH, FSH, and GPR54 Receptor Ligands 2008 17 102 49%
Synthesis of orally active small-molecule gonadotropin-releasing hormone antagonists 2004 1 34 91%
Peptidomimetic GnRH receptor antagonists for the treatment of reproductive and proliferative diseases 2006 2 73 62%
Lead compounds discovered from libraries: Part 2 2003 48 97 6%
Clinically validated peptides as templates for de novo peptidomimetic drug design at G-protein-coupled receptors 2003 30 66 8%
Gonadotropin-releasing-hormone-receptor antagonists 2001 163 96 1%

Address terms



Rank Address term Relevance score
(tfidf)
Class's shr.
of term's tot.
occurrences
Shr. of publ.
in class containing
term
Num. of
publ.
in class
1 EXPLORATORY DISCOVERY 11 69% 5.9% 9
2 STRATEG PROD PLANNING 1 19% 2.0% 3
3 ASSAY DEV GRP 0 33% 0.7% 1
4 CHEM SCREEING SCI 0 33% 0.7% 1
5 DISCOVERY PRECLIN DEV 0 25% 0.7% 1
6 PFIZER GLOBAL DEV LA JOLLA 0 25% 0.7% 1
7 HBEREICH 11 2 0 20% 0.7% 1
8 AGOURON PHARMACEUT INC 0 17% 0.7% 1
9 MEDICINAL CHEM 0 17% 0.7% 1
10 WYETH AYERST 0 14% 0.7% 1

Related classes at same level (level 1)



Rank Relatedness score Related classes
1 0.0000163646 AZALINE B//ANTIOVULATORY ACTIVITY//LHRH ANTAGONISTS
2 0.0000119465 LHRH RECEPTOR//AN 152//ENDOCRINE POLYPEPTIDE CANC
3 0.0000109108 POTENT ANTIMICROBIALS//UREA THIOUREA//3 OXAZINES
4 0.0000104644 BIOCHEM TECHNOL SCI TECHNOL//GPR35//RESONANT WAVEGUIDE GRATING BIOSENSOR
5 0.0000082073 1 4 5 6 TETRAHYDROPYRIDAZINE//BOTELL//COMBINATORIAL PARALLEL SYNTH
6 0.0000074053 4 2 THIENYLBUTYRIC ACID//SEZ CHIM FARMACEUT P PRATESI//CARBOXYAMIDATION
7 0.0000074004 PHARMACOPERONE//MOL PHARMACOL GRP//BRET
8 0.0000068983 TERMINAL NERVE//NERVUS TERMINALIS//GONADOTROPIN RELEASING HORMONE
9 0.0000068288 FUNCTIONALIZED PIPERIDINES//TETRAHYDROPYRIDINES//POLYSUBSTITUTED PIPERIDINE
10 0.0000066151 4 FLUOROPYRIMIDINES//BE CYCLES//ELE OCHEM ENERGET